Thiazesim is a benzothiazepine compound with a thiophene structure and acts as a GABAA receptor inhibitor, exerting anticonvulsant and antidepressant effects. Thiazesim exhibits specific pharmacological properties in animal experiments. Thiazesim reduces motor activity in rats and effectively inhibits rat killing responses, with a ratio of 2.1 between the ED50 in rotarod tests and the ED50 for anti-killing behavior. Thiazesim can be widely used in basic and clinical studies related to epilepsy[1][2].
Molecular Weight:
326.46
CAS Number:
[5845-26-1]
Formula:
C19H22N2OS
Target:
GABA Receptor
Application Notes:
MCE Product type: Reference compound
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